Conjugation of haloperidol to PEG allows peripheral localisation of haloperidol and eliminates CNS extrapyramidal effects
Az Alddien Natfji, D. O. Nikitin, И. И. Семина, Rouslan I. Moustafine, Vitaliy V. Khutoryanskiy, Hong Lin, Gary J. Stephens, Kimberly A. Watson, Helen M. I. Osborn, Francesca Greco
Topics & Concepts
HaloperidolCatalepsyConjugateChemistryPharmacologyIn vivoPEG ratioBlood–brain barrierReceptorBiophysicsBiochemistryDopamineEndocrinologyBiologyCentral nervous systemEconomicsBiotechnologyMathematical analysisMathematicsFinanceReceptor Mechanisms and SignalingNeuropeptides and Animal PhysiologyNeuroscience and Neuropharmacology Research