Litcius/Paper detail

Bifunctional degraders of cyclin dependent kinase 9 (CDK9): Probing the relationship between linker length, properties, and selective protein degradation

Robert J. Tokarski, Chia M. Sharpe, Andrew C. Huntsman, Brittney K. Mize, Oluwatosin R. Ayinde, Emily Stahl, James R. Lerma, Andrew Reed, Bridget Carmichael, Natarajan Muthusamy, John C. Byrd, James R. Fuchs

2023European Journal of Medicinal Chemistry25 citationsDOIOpen Access PDF

Topics & Concepts

LinkerChemistryCyclin-dependent kinaseUbiquitin ligaseKinaseUbiquitinProtein degradationBiochemistrySmall moleculeCell cycleCellGeneOperating systemComputer scienceProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsUbiquitin and proteasome pathways