Benzothiazole Amides as TRPC3/6 Inhibitors for Gastric Cancer Treatment
Yingjie Wei, Mengxian Zhang, Zhenbin Lyu, Guolin Yang, Tian Tian, Mingmin Ding, Xiaodong Zeng, Fuchun Xu, Pengyu Wang, Fangfang Li, Yixuan Liu, Zhengyu Cao, Jing Lu, Xuechuan Hong, Hongbo Wang
Abstract
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Topics & Concepts
BenzothiazoleChemistryIC50AmideTRPC6Docking (animal)AntagonistStereochemistryLead compoundPharmacologyCombinatorial chemistryReceptorIn vitroTransient receptor potential channelBiochemistryMedicineNursingIon Channels and ReceptorsBioactive Compounds and Antitumor AgentsPhytochemicals and Antioxidant Activities