Chemo-proteomics exploration of HDAC degradability by small molecule degraders
Yuan Xiong, Katherine A. Donovan, Nicholas A. Eleuteri, Nadia Kirmani, Hong Yue, Anthony Razov, Noah M. Krupnick, Radosław P. Nowak, Eric S. Fischer
Topics & Concepts
Ubiquitin ligaseChromatinProtein degradationUbiquitinHistone deacetylaseProteomicsEpigeneticsSmall moleculeHistoneProteasomeComputational biologyChromatin remodelingBiologyCell biologyChemistryBiochemistryDNAGeneProtein Degradation and InhibitorsHistone Deacetylase Inhibitors ResearchUbiquitin and proteasome pathways