New dual ATP-competitive inhibitors of bacterial DNA gyrase and topoisomerase IV active against ESKAPE pathogens
Martina Durcik, Ákos Nyerges, Žiga Skok, Darja Gramec Skledar, Jurij Trontelj, Nace Zidar, Janez Ilaš, Anamarija Zega, Cristina D. Cruz, Päivi Tammela, M. Welin, Yengo Raymond Kimbung, Dorota Focht, Ondřej Benek, Tamás Révész, Gábor Draskovits, Petra Szili, Lejla Daruka, Csaba Pál, D. Kikelj, Lucíja Peterlin Mašič, Tihomir Tomašič
Topics & Concepts
DNA gyraseTopoisomerase IVTopoisomeraseChemistryMicrobiologyDNAAntimicrobialMultiple drug resistanceBacteriaMutantMode of actionEscherichia coliBiochemistryAntibioticsBiologyGeneticsGeneCancer therapeutics and mechanismsAntibiotic Resistance in BacteriaBioactive Compounds and Antitumor Agents