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α-naphthoflavone-derived cytochrome P450 (CYP)1B1 degraders specific for sensitizing CYP1B1-mediated drug resistance to prostate cancer DU145: Structure activity relationship

Peng Chen, Shaobing Wang, Chenyang Cao, Wenchong Ye, Meizhu Wang, Cui Zhou, Wen-Ming Chen, Xu Zhang, Keyu Zhang, Wen Zhou

2021Bioorganic Chemistry17 citationsDOI

Topics & Concepts

DU145ChemistryCYP1B1Cytochrome P450PharmacologyDrug resistanceBiochemistryStereochemistryProstate cancerCancerBiologyEnzymeGeneticsLNCaPProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsUbiquitin and proteasome pathways
α-naphthoflavone-derived cytochrome P450 (CYP)1B1 degraders specific for sensitizing CYP1B1-mediated drug resistance to prostate cancer DU145: Structure activity relationship | Litcius