Litcius/Paper detail

Computational Design of Potent D-Peptide Inhibitors of SARS-CoV-2

Pedro A. Valiente, Han Wen, Satra Nim, JinAh Lee, Hyeon Ju Kim, Jinhee Kim, Albert Perez‐Riba, Yagya Prasad Paudel, Insu Hwang, Kyun‐Do Kim, Seungtaek Kim, Philip M. Kim

2021Journal of Medicinal Chemistry65 citationsDOIOpen Access PDF

Abstract

. These potent D-peptide inhibitors are promising lead candidates for developing SARS-CoV-2 prophylactic or therapeutic treatments.

Topics & Concepts

ImmunogenicityChemistryPeptidomimeticPeptideVero cellIC50In vitroSevere acute respiratory syndrome coronavirus 2 (SARS-CoV-2)AntibodyPeptide libraryVirologyReceptorBiochemistryPeptide sequenceCoronavirus disease 2019 (COVID-19)ImmunologyBiologyMedicineGeneInfectious disease (medical specialty)DiseasePathologySARS-CoV-2 and COVID-19 ResearchMonoclonal and Polyclonal Antibodies ResearchChemical Synthesis and Analysis