Discovery of baicalein derivatives as novel inhibitors against human pancreatic lipase: Structure-activity relationships and inhibitory mechanisms
Xiaoya Qin, Rong Zhu, Xu-Dong Hou, Guanghao Zhu, Min Zhang, Yufan Fan, Shenglan Qi, Jian Huang, Hui Tang, Ping Wang, Guang-Bo Ge
Topics & Concepts
BaicaleinPancreatic lipaseInhibitory postsynaptic potentialChemistryLipaseBiochemistryStructure–activity relationshipPharmacologyEnzymeBiologyIn vitroNeuroscienceFlavonoids in Medical ResearchNatural Antidiabetic Agents StudiesPhytochemicals and Antioxidant Activities