Litcius/Paper detail

Characterization of covalent binding of tyrosine kinase inhibitors to plasma proteins

Xiaoyun Liu, Dan Feng, Mingyue Zheng, Yongmei Cui, Dafang Zhong

2020Drug Metabolism and Pharmacokinetics31 citationsDOI

Topics & Concepts

Covalent bondHuman serum albuminChemistryPlasma protein bindingResidue (chemistry)MoietyBinding siteBiochemistryStereochemistryOrganic chemistryChronic Myeloid Leukemia TreatmentsChronic Lymphocytic Leukemia ResearchMonoclonal and Polyclonal Antibodies Research