Pharmacological significance of nitrogen-containing five and six-membered heterocyclic scaffolds as potent cholinesterase inhibitors for drug discovery
Rami J. Obaid, Ehsan Ullah Mughal, Nafeesa Naeem, Munirah M. Al‐Rooqi, Amina Sadiq, Rabab S. Jassas, Ziad Moussa, Saleh A. Ahmed
Topics & Concepts
ButyrylcholinesteraseAcetylcholinesteraseCholinesteraseChemistryPharmacologyCholinergicAcetylcholineEnzymeDrug discoveryDrugGalantamineAchéBiochemistryDiseaseMedicineDonepezilInternal medicineDementiaCholinesterase and Neurodegenerative DiseasesSynthesis and biological activitySynthesis and Biological Evaluation