Litcius/Paper detail

Novel antiproliferative agents bearing substituted thieno[2,3-d]pyrimidine scaffold as dual VEGFR-2 and BRAF kinases inhibitors and apoptosis inducers; design, synthesis and molecular docking

Rasha A. Hassan, Mohammed I.A. Hamed, Amr M. Abdou, Yara El‐Dash

2022Bioorganic Chemistry30 citationsDOI

Topics & Concepts

ApoptosisChemistryPyrimidineIC50KinaseSorafenibPharmacologyStereochemistryIn vitroCancer researchBiochemistryMedicineHepatocellular carcinomaSynthesis and biological activityCytokine Signaling Pathways and InteractionsCancer Mechanisms and Therapy