Pan-RAS inhibitors: Hitting multiple RAS isozymes with one stone
Alexander B. Coley, Antonio Ward, Adam B. Keeton, Xi Chen, Yulia Maxuitenko, Aishwarya Prakash, Feng Li, Jeremy B. Foote, Donald J. Buchsbaum, Gary A. Piazza
Topics & Concepts
KRASNeuroblastoma RAS viral oncogene homologHRASPopulationIsozymeCancer researchMutationCarcinogenesisBiologyCancerGeneticsMedicineGeneEnzymeBiochemistryEnvironmental healthPI3K/AKT/mTOR signaling in cancerProtein Degradation and InhibitorsProtein Kinase Regulation and GTPase Signaling