Design, synthesis and biological evaluation of dual HDAC and VEGFR inhibitors as multitargeted anticancer agents
Xue Xia, Yingjie Zhang, Yongxiang Liao, Deqing Sun, Lina Li, Ying Liu, Yongjie Wang, Wen Jiang, Jian Zhang, Yun Luan, Xiaogang Zhao
Topics & Concepts
PazopanibHDAC1PharmacologyVorinostatHistone deacetylaseHistone deacetylase inhibitorHuman umbilical vein endothelial cellChemistryHydroxamic acidUmbilical veinHDAC6Cancer researchBiologyBiochemistryCancerSunitinibHistoneIn vitroStereochemistryGeneticsGeneHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsSynthetic Organic Chemistry Methods