Development of submicromolar 17β-HSD10 inhibitors and their in vitro and in vivo evaluation
Ondřej Benek, Michaela Hanzlova, Marketa Miskerikova, Monika Schmidt, Rudolf Andrýs, Aneta Rotterova, Adam Skarka, Jana Hatlapatková, Jana Žďárová Karasová, Matej Medvecký, Lukáš Hroch, Lucie Vinklářová, Zdeněk Fišar, Jana Hroudová, Jiří Handl, Jan Čapek, Tomáš Roušar, Tereza Kobrlová, Rafael Doležal, Ondřej Soukup, Laura Aitken, Frank J. Gunn‐Moore, Kamil Musílek
Topics & Concepts
In vivoChemistryPharmacokineticsPharmacologyBioavailabilityIn vitroIC50EnzymeDrugStructure–activity relationshipBiochemistryBiologyBiotechnologyHormonal Regulation and HypertensionEstrogen and related hormone effectsATP Synthase and ATPases Research