Litcius/Paper detail

Innovative therapies for invasive fungal infections in preclinical and clinical development

Yidong Yu, Krystyna Albrecht, Jürgen Gröll, Andreas Beilhack

2020Expert Opinion on Investigational Drugs14 citationsDOI

Abstract

ABSTRACT Introduction The incidence of life-threatening invasive fungal infections (IFIs) has increased significantly in recent years. Current therapeutic options for IFIs are limited. Only four major classes of antifungal agents are available to clinicians, namely polyenes, azoles, echinocandins, and flucytosine. These antifungals have particular drawbacks, including toxicity, drug-drug interactions, and increasing antifungal resistance. Consequently, there is an urgent need for new antifungals to combat IFIs. Areas covered This review illuminates new classes of synthetic antifungal drugs under preclinical and clinical investigations that have novel mechanisms of action; it also examines innovative strategies for the in vivo delivery of antifungal drugs. Expert opinion It is imperative to expand the pipeline of antifungals to tackle emerging fungal resistance against conventional antimycotic drugs, toxicity, and drug-drug interactions. This unmet medical need should not be underappreciated.

Topics & Concepts

EchinocandinsFlucytosineAntifungalDrugAntifungal drugsMedicineIntensive care medicineAntifungal drugPharmacologyDrug resistanceClinical trialAmphotericin BBiologyInternal medicineCaspofunginMicrobiologyDermatologyAntifungal resistance and susceptibilityFungal Infections and StudiesNail Diseases and Treatments