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CDK4/6 inhibitors: a brief overview and prospective research directions

Tenzin Adon, Dhivya Shanmugarajan, Honnavalli Yogish Kumar

2021RSC Advances64 citationsDOIOpen Access PDF

Abstract

In this article, we explore the biological importance of CDK4/6 in cancer therapy, the development of resistance to monotherapy, and a short overview of PROTAC (Proteolysis Targeting Chimera), a unique and pioneering technique for degrading CDK4/6 enzymes. Overall, our prime focus is to discuss novel CDK4/6 inhibitors with diverse chemical classes and their correlation with computational studies.

Topics & Concepts

PsychologyAdvanced Breast Cancer TherapiesCancer-related Molecular PathwaysCancer-related cognitive impairment studies
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