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A practical guide for the assay-dependent characterisation of irreversible inhibitors

Lavleen Mader, Jessica E. Borean, Jeffrey W. Keillor

2024RSC Medicinal Chemistry20 citationsDOIOpen Access PDF

Abstract

Kinetic evaluations for assay dependent characterization of irreversible inhibitors.

Topics & Concepts

Computational biologyComputer scienceChemistryBiologyComputational Drug Discovery MethodsMonoclonal and Polyclonal Antibodies ResearchInnovative Microfluidic and Catalytic Techniques Innovation
A practical guide for the assay-dependent characterisation of irreversible inhibitors | Litcius