Human carboxylesterase 1A plays a predominant role in the hydrolytic activation of remdesivir in humans
Feng Zhang, Hongxin Li, Tiantian Zhang, Yuan Xiong, Haonan Wang, Zhenhui Lu, Lei Xiong, Yuqi He, Guang‐Bo Ge
Topics & Concepts
CarboxylesteraseHydrolysisButyrylcholinesteraseChemistryEnzymeProdrugPharmacologyAcetylcholinesteraseBiochemistryMedicineAchéCholinesterase and Neurodegenerative DiseasesPharmaceutical Practices and Patient OutcomesComputational Drug Discovery Methods