Store-Operated Calcium Entry as a Therapeutic Target in Acute Pancreatitis: Discovery and Development of Drug-Like SOCE Inhibitors
M. Teresa Serafini, Celia Cordero-Sánchez, Rosanna Di Paola, Irene Preet Bhela, Silvio Aprile, Beatrice Purghè, Roberta Fusco, Salvatore Cuzzocrea, Armando A. Genazzani, Beatrice Riva, Tracey Pirali
Abstract
efficacy in a mouse model of acute pancreatitis.
Topics & Concepts
ChemistryIn vivoAcute pancreatitisDrugDrug discoveryPharmacologyMechanism (biology)CalciumPancreatitisHomeostasisBiochemistryCell biologyInternal medicineMedicineBiologyOrganic chemistryEpistemologyBiotechnologyPhilosophyBioactive Compounds and Antitumor AgentsCalcium signaling and nucleotide metabolismIon Channels and Receptors