Design, synthesis and biological evaluation of KRASG12C-PROTACs
Xiaoyi Zhang, Tong Zhao, Minghao Sun, Pei Li, Mengzhen Lai, Lingfeng Xie, Jiaying Chen, Jian Ding, Hua Xie, Jinpei Zhou, Huibin Zhang, Jinpei Zhou, Huibin Zhang
Topics & Concepts
ChemistryProteasomeSmall moleculeEpothilonePharmacologyBiochemistryStereochemistryBiologyProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysMultiple Myeloma Research and Treatments