Flavonoid analogues as urease inhibitors: Synthesis, biological evaluation, molecular docking studies and in-silico ADME evaluation
H. Liu, Yan Wang, Mingxia Lv, Yi Luo, Buming Liu, Yan Huang, Mian Wang, Jianyi Wang
Topics & Concepts
ChemistryUreaseDruggabilityADMEThioureaIn silicoDocking (animal)FlavonoidCombinatorial chemistryBiochemistryIC50In vitroStereochemistryEnzymePharmacologyOrganic chemistryAntioxidantGeneMedicineNursingMicrobial Applications in Construction MaterialsSynthesis and biological activitySynthesis and Characterization of Heterocyclic Compounds