Fragment-based design and synthesis of coumarin-based thiazoles as dual c-MET/STAT-3 inhibitors for potential antitumor agents
Bassem H. Naguib, Heba A. Elsebaie, Mohamed S. Nafie, Samy Mohamady, Nader R. Albujuq, Aya Samir Ayed, Dina Nada, Ahmed Khalil, Salma M. Hefny, Haytham O. Tawfik, Moataz A. Shaldam
Topics & Concepts
CoumarinChemistryIn vitroCancer cell linesStereochemistrystatCancer cellCombinatorial chemistryCancerPharmacologyApoptosisBiochemistrySTAT3Organic chemistryInternal medicineMedicineSynthesis and biological activityCytokine Signaling Pathways and InteractionsSynthesis of heterocyclic compounds