Design, synthesis and biological evaluation of novel diazaspirodecanone derivatives containing piperidine-4-carboxamide as chitin synthase inhibitors and antifungal agents
Qinggang Ji, Bing Li, Yiwen Chu, Hu Wu, Chuanbiao Du, Yajie Xu, Yangli Shen, Junfeng Deng
Topics & Concepts
ChemistryCandida albicansIC50ChitinFluconazoleCryptococcus neoformansStereochemistryPotencyMinimum inhibitory concentrationChitin synthaseATP synthaseAntifungalIn vitroEnzymeBiochemistryMicrobiologyChitosanBiologyCarbohydrate Chemistry and SynthesisStudies on Chitinases and ChitosanasesFungal Plant Pathogen Control