The impact of cryo-EM on determining allosteric modulator-bound structures of G protein-coupled receptors
Liudi Zhang, Jesse I. Mobbs, Lauren T. May, Alisa Glukhova, David M. Thal
Topics & Concepts
Allosteric regulationG protein-coupled receptorDrug discoverySmall moleculeComputational biologyAllosteric modulatorLigand (biochemistry)Structural biologyBinding siteBiologyReceptorChemistryBiophysicsNanotechnologyBioinformaticsBiochemistryMaterials scienceReceptor Mechanisms and SignalingMass Spectrometry Techniques and ApplicationsMonoclonal and Polyclonal Antibodies Research