Design, synthesis, and anti-inflammatory activity characterization of novel brain-permeable HDAC6 inhibitors
Gang Liu, Prasenjit Mondal, Na Sang, Zihua Li, Weihua Ding, Liuyue Yang, Yan Liu, Vishal C. Birar, Ashley Gomm, Rudolph E. Tanzi, Can Zhang, Shiqian Shen, Changning Wang, Xiaoxia Lü, Ping Bai
Topics & Concepts
NeuroinflammationHDAC6ChemistryMicrogliaIn vivoPharmacologyInflammationBiodistributionHistone deacetylaseIn vitroBiochemistryCancer researchImmunologyHistoneBiologyBiotechnologyGeneHistone Deacetylase Inhibitors ResearchPeptidase Inhibition and AnalysisAdenosine and Purinergic Signaling