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Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice

Elliot D. Mock, Mohammed Ahmed Mustafa, Ozge Gunduz‐Cinar, Reşat Çınar, Gavin N. Petrie, Vasudev Kantae, Xinyu Di, Daisuke Ogasawara, Zoltán V. Varga, János Pálóczi, Cristina Miliano, Giulia Donvito, Annelot C. M. van Esbroeck, Anouk M. F. van der Gracht, Ioli Kotsogianni, Joshua K. Park, Andrea Martella, Tom van der Wel, Marjolein Soethoudt, Ming Jiang, Tiemen J. Wendel, Antonius P. A. Janssen, Alexander T. Bakker, Colleen Donovan, Laura I. Castillo, Bogdan I. Florea, Jesse W.Y. Wat, Helma van den Hurk, Matthias Wittwer, Uwe Grether, Andrew Holmes, C. A. A. VAN BOECKEL, Thomas Hankemeier, Benjamin F. Cravatt, Matthew W. Buczynski, Matthew N. Hill, Pál Pacher, Aron H. Lichtman, Mario van der Stelt

2020Nature Chemical Biology96 citationsDOIOpen Access PDF

Topics & Concepts

AnandamideFatty acid amide hydrolaseEndocannabinoid systemCannabinoid receptorCannabinoidLipid signalingPhospholipase DNeuroprotectionBiologyChemistryAntagonistEndocrinologyNeuroscienceCell biologyReceptorSignal transductionBiochemistryCannabis and Cannabinoid ResearchPancreatic function and diabetesSleep and Wakefulness Research
Discovery of a NAPE-PLD inhibitor that modulates emotional behavior in mice | Litcius