Design, Synthesis, and Structure-Activity relationships of Evodiamine-Based topoisomerase (Top)/Histone deacetylase (HDAC) dual inhibitors
Fugui Zhu, Xiangguo Meng, Huixin Liang, Chunquan Sheng, Guoqiang Dong, Dan Liu, Shanchao Wu
Topics & Concepts
EvodiamineChemistryHistone deacetylaseAcetylationTopoisomeraseHDAC6ApoptosisCell cycle checkpointIn vitroTrichostatin AHistoneCell cycleBiochemistryDNAChromatographyGeneCancer therapeutics and mechanismsHistone Deacetylase Inhibitors ResearchQuinazolinone synthesis and applications