DC591017, a phosphodiesterase-4 (PDE4) inhibitor with robust anti-inflammation through regulating PKA-CREB signaling
Heng Li, Jian Li, Xianglei Zhang, Chunlan Feng, Chen Fan, Xiaoqian Yang, Rui Zhang, Fenghua Zhu, Yu Zhou, Yechun Xu, Hong Liu, Wei Tang
Topics & Concepts
CREBInflammationPhosphodiesteraseIn vivoPharmacologyGene knockdownChemistryForskolinPhosphodiesterase inhibitorSignal transductionImmunologyMedicineIn vitroBiologyTranscription factorEnzymeBiochemistryBiotechnologyGeneApoptosisMast cells and histaminePsoriasis: Treatment and PathogenesisAsthma and respiratory diseases