Safinamide's potential in treating nondystrophic myotonias: Inhibition of skeletal muscle voltage-gated sodium channels and skeletal muscle hyperexcitability in vitro and in vivo
Jean‐François Desaphy, Alessandro Farinato, Concetta Altamura, Michela De Bellis, Paola Imbrici, Nancy Tarantino, Carla Caccia, Elsa Melloni, Gloria Padoani, Silvia Vailati, Charlotte Keywood, Maria Rosaria Carratù, Annamaria De Luca, Diana Conte Camerino, Sabata Pierno
Topics & Concepts
MexiletineChemistrySodium channelSodium channel blockerPharmacologySkeletal muscleBiophysicsSodiumInternal medicineMedicineBiologyOrganic chemistryIon channel regulation and functionNeuroscience and Neural EngineeringCardiac electrophysiology and arrhythmias