Discovery of novel nucleoside derivatives as selective lysine acetyltransferase p300 inhibitors for cancer therapy
Qiuzi Dai, Zigao Yuan, Qinsheng Sun, Zhuolin Ao, Binsheng He, Yuyang Jiang
Topics & Concepts
ChemistryHistone acetyltransferaseAcetylationLysineEpigeneticsAcetyltransferaseNucleosideHistone AcetyltransferasesBiochemistryCancerCancer researchPharmacologyBiologyAmino acidGeneGeneticsGenomics and Chromatin DynamicsProtein Degradation and InhibitorsEpigenetics and DNA Methylation