Computational Modeling and Pharmacokinetics/ADMET Study of Some Arylpiperazine Derivatives as Novel Antipsychotic Agents Targeting Depression
Sabitu Babatunde Olasupo, Adamu Uzairu, Gideon Shallangwa Adamu, Sani Uba
Topics & Concepts
Quantitative structure–activity relationshipIn silicoPharmacophorePharmacokineticsChemistryhERGSerotonin transporterPharmacologyAntipsychoticComputational biologyStereochemistryBiochemistryReceptorMedicineBiologyGeneSerotoninSchizophrenia (object-oriented programming)Internal medicinePotassium channelPsychiatryComputational Drug Discovery MethodsTreatment of Major DepressionSynthesis and biological activity