Identification of new anti-mycobacterial agents based on quinoline-isatin hybrids targeting enoyl acyl carrier protein reductase (InhA)
Eman F. Khaleel, Ahmed Sabt, Małgorzata Korycka‐Machała, Rehab Mustafa Badi, Ninh The Son, Nguyen Xuan Ha, Mohamed Farouk Hamissa, Ahmed E. Elsawi, Eslam B. Elkaeed, Bożena Dziadek, Wagdy M. Eldehna, Jarosław Dziadek, Jarosław Dziadek
Topics & Concepts
INHAIsatinChemistryMycobacterium tuberculosisEnzymeIsoniazidBiochemistryReductaseDocking (animal)Active siteQuinolineStereochemistryTuberculosisMedicineNursingPathologyOrganic chemistryTuberculosis Research and EpidemiologyComputational Drug Discovery MethodsAntimicrobial agents and applications