Design, synthesis, and biological evaluation of novel discoidin domain receptor inhibitors for the treatment of lung adenocarcinoma and pulmonary fibrosis
Shangke Liu, Xiang Li, Can Chen, Xinyu Lin, Wei‐Fang Zuo, Cheng Peng, Qinglin Jiang, Wei Huang, Gu He
Topics & Concepts
Discoidin domainDDR1In vivoChemistryPharmacologyCancer researchMAPK/ERK pathwayA549 cellBleomycinDasatinibFibrosisPulmonary fibrosisReceptorKinaseIn vitroBiochemistryPathologyReceptor tyrosine kinaseMedicineBiologyTyrosine kinaseInternal medicineBiotechnologyChemotherapyCell Adhesion Molecules ResearchHER2/EGFR in Cancer ResearchMonoclonal and Polyclonal Antibodies Research