Litcius/Paper detail

Design, synthesis, and biological evaluation of novel discoidin domain receptor inhibitors for the treatment of lung adenocarcinoma and pulmonary fibrosis

Shangke Liu, Xiang Li, Can Chen, Xinyu Lin, Wei‐Fang Zuo, Cheng Peng, Qinglin Jiang, Wei Huang, Gu He

2023European Journal of Medicinal Chemistry10 citationsDOIOpen Access PDF

Topics & Concepts

Discoidin domainDDR1In vivoChemistryPharmacologyCancer researchMAPK/ERK pathwayA549 cellBleomycinDasatinibFibrosisPulmonary fibrosisReceptorKinaseIn vitroBiochemistryPathologyReceptor tyrosine kinaseMedicineBiologyTyrosine kinaseInternal medicineBiotechnologyChemotherapyCell Adhesion Molecules ResearchHER2/EGFR in Cancer ResearchMonoclonal and Polyclonal Antibodies Research