Discovery of pyrazole N-aryl sulfonate: A novel and highly potent cyclooxygenase-2 (COX-2) selective inhibitors
Haiyan Yao, Quanping Guo, Mengran Wang, Rui Wang, Zhaoqing Xu
Topics & Concepts
SulfonatePyrazoleChemistryArylIn vivoStereochemistryMedicinal chemistryOrganic chemistrySodiumBiologyBiotechnologyAlkylInflammatory mediators and NSAID effectsSynthesis and biological activitySynthesis and Biological Evaluation