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Optimization of bifunctional piperidinamide derivatives as σ1R Antagonists/MOR agonists for treating neuropathic pain

Jiaying Xiong, Tao Zhuang, Yurong Ma, Junyi Xu, Jiaqi Ye, Ru Ma, Shuang Zhang, Xin Liu, Bi‐Feng Liu, Chao Hao, Guisen Zhang, Yin Chen

2021European Journal of Medicinal Chemistry22 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryNeuropathic painAnalgesicPharmacologyOpioidSedationStereochemistryAnesthesiaReceptorMedicineBiochemistryPharmacological Receptor Mechanisms and EffectsNeuropeptides and Animal PhysiologyPain Mechanisms and Treatments
Optimization of bifunctional piperidinamide derivatives as σ1R Antagonists/MOR agonists for treating neuropathic pain | Litcius