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A novel potent metal-binding NDM-1 inhibitor was identified by fragment virtual, SPR and NMR screening

Huifang Guo, Kai Cheng, Yan Gao, Weiqi Bai, Cai Wu, Wei He, Conggang Li, Zhuorong Li

2020Bioorganic & Medicinal Chemistry20 citationsDOI

Topics & Concepts

ChemistryVirtual screeningPharmacophoreStereochemistryCombinatorial chemistryAntibacterial activityBacteriaBiologyGeneticsAntibiotic Resistance in BacteriaPneumocystis jirovecii pneumonia detection and treatmentTuberculosis Research and Epidemiology
A novel potent metal-binding NDM-1 inhibitor was identified by fragment virtual, SPR and NMR screening | Litcius