Optimising proteolysis-targeting chimeras (PROTACs) for oral drug delivery: a drug metabolism and pharmacokinetics perspective
Andy Pike, Beth Williamson, Stephanie Harlfinger, Scott Martin, Dermot F. McGinnity
Topics & Concepts
PharmacokineticsDrugDrug discoveryDrug metabolismPharmacologyMedicineComputational biologyBioinformaticsBiologyProtein Degradation and InhibitorsPeptidase Inhibition and AnalysisUbiquitin and proteasome pathways