High-throughput fluorescent screening of thioredoxin reductase inhibitors to inhibit Mycobacterium tuberculosis
Fei Yan, Xin Zhao, Ruibo Li, Xiuyan Han, Qiulong Yan, Lei Feng, Xiulan Xin, Jingnan Cui, Xiaochi Ma
Topics & Concepts
Mycobacterium tuberculosisDrug discoveryThioredoxin reductaseTuberculosisPathogenChemistryDrugMicrobiologyReductaseThioredoxinBiologyBiochemistryEnzymePharmacologyMedicinePathologySynthesis and biological activityComputational Drug Discovery MethodsEnzyme function and inhibition