Heteroarene-fused anthraquinone derivatives as potential modulators for human aurora kinase B
Mandeep Singh, Lakshay Malhotra, Md. Anzarul Haque, Mukesh Kumar, Alexander S. Tikhomirov, Valeria A. Litvinova, Alexander M. Korolev, A.S. Ethayathulla, Uddipan Das, Andrey E. Shchekotikhin, Punit Kaur
Topics & Concepts
ChemistryAurora kinaseKinaseIn silicoPharmacophoreVirtual screeningIn vitroAurora B kinaseMoietyAurora inhibitorComputational biologyBiochemistryPharmacologyStereochemistryBiologyCellCell divisionSpindle apparatusCell cycleGeneMicrotubule and mitosis dynamicsProtein Degradation and Inhibitors14-3-3 protein interactions