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An EDA complex-driven multicomponent reaction of Br–R <sub>f</sub> with alkenes <i>via</i> radical-polar crossover

Zhen Chen, Jin-Xin Lan, Shupeng Zhang, SM Lu, Yicheng Zhang, Wenchao Yang

2025Chemical Communications12 citationsDOI

Abstract

, offering a mild, operationally simple, and broadly applicable alternative to traditional post modification of nitrogen heterocycles. This reaction involved a cascade XAT/radical addition/radical polar crossover/radical addition to nitrogen heterocycles/HAT process.

Topics & Concepts

CascadeNitrogenChemistryCrossoverReaction conditionsCascade reactionCombinatorial chemistryPolarComputational chemistryOrganic chemistryReaction mechanismMaterials scienceNanotechnologySurface modificationComponent (thermodynamics)Reaction intermediateRadical Photochemical ReactionsCatalytic C–H Functionalization MethodsCatalytic Cross-Coupling Reactions
An EDA complex-driven multicomponent reaction of Br–R <sub>f</sub> with alkenes <i>via</i> radical-polar crossover | Litcius