Discovery of novel Staphylococcus aureus penicillin binding protein 2a inhibitors by multistep virtual screening and biological evaluation
Na Lv, Qinxiang Kong, Hui Zhang, Jiabin Li
Topics & Concepts
Staphylococcus aureusChemistryPenicillin binding proteinsVirtual screeningPenicillinAntibacterial agentDrug discoveryMicrobiologyBiological activityMicrococcaceaeAntibioticsBacteriaComputational biologyCombinatorial chemistryIn vitroBiochemistryBiologyGeneticsAntimicrobial Resistance in StaphylococcusBiochemical and Structural CharacterizationMonoclonal and Polyclonal Antibodies Research