Design and synthesis of anti–inflammatory 1,2,3–triazolylpyrrolobenzodiazepinone derivatives and impact of molecular structure on COX–2 selective targeting
Amit Kumar, Mohammad Sarwar Alam, Hinna Hamid, Vaishali Chugh, Tanvi Tikla, Rajeev Kaul, Abhijeet Dhulap, Sunil Sharma
Topics & Concepts
ChemistryCelecoxibIn vivoPharmacologyIn silicoEnzymeIn vitroDrug discoveryDrugIC50HeLaStructure–activity relationshipArachidonic acidAnti-inflammatoryBiochemistryStereochemistryMedicineBiotechnologyBiologyGeneClick Chemistry and ApplicationsSynthesis and Biological EvaluationSynthesis of β-Lactam Compounds