Half-life extension of peptidic APJ agonists by N-terminal lipid conjugation
Anthony B. Reed, Brian A. Lanman, Jerry Ryan Holder, Bryant H. Yang, Ji Ma, Sara C. Humphreys, Zhican Wang, Joyce Chan, Les P. Miranda, Gayathri Swaminath, John G. Allen
Topics & Concepts
ChemistryApelinAgonistReceptorInotropeAngiotensin IIAngiotensin II receptor type 1PharmacologyInternal medicineEndogenous agonistEndocrinologyPeptideBiochemistryBiologyMedicineDopamine receptor D1Apelin-related biomedical researchCardiovascular, Neuropeptides, and Oxidative Stress ResearchHormonal Regulation and Hypertension