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Accelerated rational PROTAC design via deep learning and molecular simulations

Shuangjia Zheng, Youhai Tan, Zhenyu Wang, Chengtao Li, Zhiqing Zhang, Xu Sang, Hongming Chen, Yuedong Yang

2022Nature Machine Intelligence141 citationsDOIOpen Access PDF

Topics & Concepts

BromodomainComputer scienceArtificial intelligenceDeep learningRational designComputational biologyMachine learningBiologyNanotechnologyMaterials scienceBiochemistryGeneAcetylationProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysMultiple Myeloma Research and Treatments
Accelerated rational PROTAC design via deep learning and molecular simulations | Litcius