Oxa-376 and Oxa-530 variants of β-lactamase: computational study uncovers potential therapeutic targets of<i>Acinetobacter baumannii</i>
Sajal Kumar Halder, Maria Mulla Mim, Md. Meharab Hassan Alif, Jannatul Fardous Shathi, Nuhu Alam, Aparna Shil, Mahbubul Kabir Himel
Abstract
Determining novel therapeutic targets of Acinetobacter baumannii . Deleterious variants, causing antibiotic resistance, were identified by molecular docking and molecular dynamics simulation suggesting new therapeutic targets Oxa-376 and Oxa-530.
Topics & Concepts
Acinetobacter baumanniiMultiple drug resistanceAntibiotic resistanceAntimicrobialMicrobiologyBacteriaMutantDrug resistanceComputational biologyAntibioticsBiologyChemistryGeneticsPseudomonas aeruginosaGeneAntibiotic Resistance in BacteriaCancer therapeutics and mechanismsBerberine and alkaloids research