Quinoline carboxamide core moiety-based compounds inhibit P. falciparumfalcipain-2: Design, synthesis and antimalarial efficacy studies
Anju Singh, Md Kalamuddin, Mudasir Maqbool, Asif Mohmmed, Pawan Malhotra, Nasimul Hoda
Topics & Concepts
ChemistryQuinolineIn silicoPharmacologyAntimalarial AgentMoietyPlasmodium falciparumCysteine proteaseCarboxamideIn vitroBiochemistryCombinatorial chemistryStereochemistryMalariaProteaseEnzymeBiologyOrganic chemistryGeneImmunologyMalaria Research and ControlComputational Drug Discovery MethodsResearch on Leishmaniasis Studies