Synthesis and pharmacokinetic study of a 11C-labeled cholesterol 24-hydroxylase inhibitor using ‘in-loop’ [11C]CO2 fixation method
Zhen Chen, Jiahui Chen, Natalia Mast, Jian Rong, Xiaoyun Deng, Tuo Shao, Hualong Fu, Qingzhen Yu, Jiyun Sun, Yihan Shao, Lee Josephson, Thomas Collier, Irina A. Pikuleva, Steven H. Liang
Topics & Concepts
ChemistryMetaboliteCytochrome P450MonooxygenasePharmacokineticsCholesterolEnzymeEnzyme inhibitorPharmacologyBiochemistryBiologyHormonal Regulation and HypertensionCholesterol and Lipid MetabolismSteroid Chemistry and Biochemistry