Litcius/Paper detail

Synthesis and pharmacokinetic study of a 11C-labeled cholesterol 24-hydroxylase inhibitor using ‘in-loop’ [11C]CO2 fixation method

Zhen Chen, Jiahui Chen, Natalia Mast, Jian Rong, Xiaoyun Deng, Tuo Shao, Hualong Fu, Qingzhen Yu, Jiyun Sun, Yihan Shao, Lee Josephson, Thomas Collier, Irina A. Pikuleva, Steven H. Liang

2020Bioorganic & Medicinal Chemistry Letters11 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryMetaboliteCytochrome P450MonooxygenasePharmacokineticsCholesterolEnzymeEnzyme inhibitorPharmacologyBiochemistryBiologyHormonal Regulation and HypertensionCholesterol and Lipid MetabolismSteroid Chemistry and Biochemistry