Litcius/Paper detail

Design, synthesis and antitumor activity study of PARP-1/HDAC dual targeting inhibitors

Ziwei Chi, Ying Bai, Jing Li, KeWei Wang, Yungen Xu, Yepeng Luan

2022Bioorganic & Medicinal Chemistry Letters24 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryAcetylationHistone deacetylasePoly ADP ribose polymeraseHDAC6OlaparibPARP inhibitorBenzimidazoleCancer researchCell growthPharmacologyHistoneBiochemistryPolymeraseEnzymeBiologyDNAOrganic chemistryGenePARP inhibition in cancer therapyHistone Deacetylase Inhibitors ResearchSignaling Pathways in Disease
Design, synthesis and antitumor activity study of PARP-1/HDAC dual targeting inhibitors | Litcius