Structure-guided optimization of adenosine mimetics as selective and potent inhibitors of coronavirus nsp14 N7-methyltransferases
Marcel Hausdorff, Adrien Delpal, Sarah Barelier, Laura Nicollet, Bruno Canard, Franck Touret, Agathe M. G. Colmant, Bruno Coutard, Jean‐Jacques Vasseur, Étienne Decroly, Françoise Debart
Topics & Concepts
ChemistryMethyltransferaseAdenosineCoronavirusStereochemistryBiochemistryCoronavirus disease 2019 (COVID-19)MethylationGeneInternal medicineDiseaseInfectious disease (medical specialty)MedicineRNA modifications and cancerTuberculosis Research and EpidemiologyRNA Interference and Gene Delivery