Litcius/Paper detail

PLK1 (polo like kinase 1)-dependent autophagy facilitates gefitinib-induced hepatotoxicity by degrading COX6A1 (cytochrome c oxidase subunit 6A1)

Peihua Luo, Hao Yan, Jiangxia Du, Xueqin Chen, Jinjin Shao, Ying Zhang, Zhifei Xu, Ying Jin, Nengming Lin, Bo Yang, Qiaojun He

2020Autophagy78 citationsDOIOpen Access PDF

Abstract

3-MA: 3-methyladenine; AAV8: adeno-associated virus serotype 8; ATG5: autophagy related 5; ATG7: autophagy related 7; B2M: beta-2-microglobulin; CCCP: carbonyl cyanide m-chlorophenylhydrazone; CHX: cycloheximide; COX6A1: cytochrome c oxidase subunit 6A1; c-PARP: cleaved poly(ADP-ribose) polymerase; CQ: chloroquine; GOT1/AST: glutamic-oxaloacetic transaminase 1, soluble; GPT/ALT: glutamic pyruvic transaminase, soluble; HBSS: Hanks´ balanced salt solution; H&E: hematoxylin and eosin; MAP1LC3/LC3: microtubule associated proteins 1 light chain 3; PLK1: polo like kinase 1; RCC IV: respiratory chain complex IV; ROS: reactive oxygen species; TUBB8: tubulin beta 8 class VIII.

Topics & Concepts

GefitinibAutophagyBiologyCancer researchEpidermal growth factor receptorApoptosisATG5CancerBiochemistryGeneticsAutophagy in Disease and TherapyPI3K/AKT/mTOR signaling in cancerQuinazolinone synthesis and applications